Research Focus
Technology Platforms & Research Areas
Our scientific team is actively engaged across the following technology platforms and research areas.
Peptide Chemistry
Solid-Phase Peptide Synthesis
- • Fmoc/Boc strategies
- • Automated & manual synthesis
- • Difficult sequence optimization
Cyclic & Constrained Peptides
- • Head-to-tail cyclization
- • Stapled peptides
- • Disulfide-constrained scaffolds
Peptide-Drug Conjugates
- • Targeted delivery peptides
- • Linker-payload optimization
- • Stability & PK studies
Medicinal Chemistry
Structure-Activity Relationship (SAR) Studies
- • Analog design
- • Potency optimization
- • Selectivity profiling
Small-Molecule Lead Optimization
- • ADMET-guided design
- • Scaffold hopping
- • Synthetic route scouting
Fragment-Based Design
- • Fragment library synthesis
- • Hit-to-lead expansion
- • Crystallography-guided design
Bioconjugation
Antibody-Drug Conjugates (ADC)
- • Site-specific conjugation
- • Linker chemistry
- • DAR characterization
Click Chemistry & Bioorthogonal Labeling
- • SPAAC/CuAAC methods
- • Bioorthogonal handles
- • In-vivo labeling strategies
PEGylation & Half-Life Extension
- • PEG linker selection
- • Site-specific PEGylation
- • Pharmacokinetic evaluation
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